|
SHR
|
SHR/H
|
SHR-mtBN
|
SHR-mtBN/H
|
---|
B
max (fmol mg−1)
|
21.71 ± 0.88
|
25.20 ± 0.38+
|
24.87 ± 0.73
|
18.37 ± 0.46§#
|
K
D (nM)
|
0.49 ± 0.10
|
0.58 ± 0.07
|
0.51 ± 0.03
|
0.32 ± 0.01
|
- Data are means (±SEM) of three separate experiments performed in triplicates
-
B
max
maximal binding capacity, K
D
equilibrium dissociation constant of radioligand ([3H]CGP 12177)
-
+
p < 0.05 SHR vs. SHR/H; § p < 0.05 SHR/H vs. SHR-mtBN/H rats; # p < 0.05 SHR-mtBN vs. SHR-mtBN/H